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Tabimorelin Hemifumarate, Potent, Orally Active Ghrelin Receptor Agonist, Each

632.48

Details:

Potent, orally active ghrelin receptor (GHS-R1a) agonist (Ki = 50 nM at human recombinant GHS-R1a). Stimulates GH release from rat pituitary cells with an EC50 value of 2.7 nM. Induces hyperphagia and adiposity in lean rats, but not in leptin signaling-deficient ZDF rats.

Additional Information

SKU 10455163
UOM Each
UNSPSC 12352200
Manufacturer Part Number 2308/10