Mrs 5698, High Affinity And Selective A3 Agonist, Each

Details:

Mrs 5698 is a high affinity and selective a3 adenosine receptor agonist (ki ∽ 3 nm); displays >1000-fold selectivity over a1 and a2a adenosine receptors. Reverses mechanoallodynia in several neuropathic pain models in vivo. Orally bioavailable.